Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
G protein-coupled receptor 119 (Macaca fascicularis) | BDBM50445481 (CHEMBL3104879) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 73 | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Agonist activity at cynomolgus monkey GPR119 assessed as cAMP accumulation | Bioorg Med Chem Lett 24: 156-60 (2013) Article DOI: 10.1016/j.bmcl.2013.11.053 BindingDB Entry DOI: 10.7270/Q2J104N3 | |||||||||||
More data for this Ligand-Target Pair |