Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133685 (CHEMBL3633663) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133685 (CHEMBL3633663) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133679 (CHEMBL3633665) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133679 (CHEMBL3633665) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133682 (CHEMBL3633656) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133682 (CHEMBL3633656) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133681 (CHEMBL3633655) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.13E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133681 (CHEMBL3633655) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.14E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133676 (CHEMBL3633650) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133676 (CHEMBL3633650) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133677 (CHEMBL3633651) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.98E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133677 (CHEMBL3633651) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.98E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133686 (CHEMBL3633664) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.73E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133686 (CHEMBL3633664) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.75E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133680 (CHEMBL3633654) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.61E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133680 (CHEMBL3633654) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.61E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133678 (CHEMBL3633653) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.32E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133678 (CHEMBL3633653) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.32E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133683 (CHEMBL3633657) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.45E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133683 (CHEMBL3633657) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.48E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133684 (CHEMBL3633662) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.56E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133684 (CHEMBL3633662) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.57E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133688 (CHEMBL3633658) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133689 (CHEMBL3633659) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133690 (CHEMBL3633660) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133691 (CHEMBL3633661) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor family C group 6 member A (Mus musculus) | BDBM50133687 (CHEMBL3633652) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at mouse GPRC6A receptor expressed in HEK293 cells assessed as inhibition of L-ornithine-induced inositol monophosphate accumulat... | J Med Chem 58: 8938-51 (2015) Article DOI: 10.1021/acs.jmedchem.5b01254 BindingDB Entry DOI: 10.7270/Q2DF6T1G | |||||||||||
More data for this Ligand-Target Pair |