Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396227 (6-[5-Bromo-6-(2-oxa-6-aza-spiro[3.3]hept-6-yl)-pyr...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0200 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396236 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0200 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396236 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.0200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISA | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396194 (6-(5-Bromo-6-methoxy-pyridin-2-ylmethyl)-5-methyl-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0220 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396205 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0260 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396220 (6-(5-Bromo-6-morpholin-4-yl-pyridin-2-ylmethyl)-5-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0260 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396239 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0270 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396246 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0270 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM50548078 (CHEMBL4746798) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.0280 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISA | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396118 (6-(5,6-Dibromo-pyridin-2-ylmethyl)-5-methyl-[1,2,5...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0300 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396219 (1-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0330 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396233 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0330 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396197 (6-[5-Bromo-6-(2-fluoro-ethoxy)-pyridin-2-ylmethyl]...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0340 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396222 (6-(5-Bromo-6-cyclopropylamino-pyridin-2-ylmethyl)-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0380 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396112 (6-(6-Bromo-5-difluoromethoxy-pyridin-2-ylmethyl)-5...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0380 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396218 (6-{5-Bromo-6-[(3-methyl-oxetan-3-ylmethyl)-amino]-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0450 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396240 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0460 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396116 (6-(5-Brom32.2-chloro-pyridin-2-ylmethyl)-5-methyl-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0470 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396164 (6-(6-Amino-5-thiazol-5-yl-pyridin-2-ylmethyl)-5-me...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0500 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396226 (6-[5-Bromo-6-(3,3-difluoro-azetidin-1-yl)-pyridin-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0520 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396234 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0540 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396241 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0550 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396221 (3-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0560 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396189 (6-[5-Bromo-6-(2,2-difluoro-ethoxy)-pyridin-2-yl me...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0580 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396191 (1-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0580 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM50548079 (CHEMBL4754865) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.0660 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISA | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396119 (6-(5-Brom32.2-fluoro-pyridin-2-ylmethyl)-5-methyl-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0660 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396196 (6-[5-Bromo-6-(2,2-difluoro-propoxy)-pyridin-2-ylme...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0720 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396139 (6-(7-amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0730 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396198 (6-[5-Bromo-6-(3-fluoro-propoxy)-pyridin-2-yl methy...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0740 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396199 (6-(5-Bromo-6-methylsulfanyl-pyridin-2-ylmethyl)-5-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0740 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396235 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0750 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396180 (6-[5-bromo-4-(trifluoromethyl)pyrimidin-2-yl]methy...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0770 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396193 (6-[5-Bromo-6-(2,2,2-trifluoro-ethoxy)-pyridin-2-yl...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0790 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396120 (6-(5-Brom32.2-difluoromethoxy-pyridin-2-ylmethyl)-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0820 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396167 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0820 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396192 (6-[5-Bromo-6-(3-methyl-oxetan-3-ylmethoxy)-pyridin...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0820 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396215 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0850 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396200 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0860 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396216 (6-(6-Amino-5-difluoromethoxy-pyridin-2-ylmethyl)-5...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0910 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396206 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0930 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396225 (6-[5-Bromo-6-(3,3-difluoro-cyclobutylamino)-pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0960 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396228 (1-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0970 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396230 (6-[5-Bromo-6-(3,3-difluoro-propylamino)-pyridin-2-...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0990 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396224 (3-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396154 (6-(6-Furan-2-yl-pyridin-2-ylmethyl)-5-methyl-[1,2,...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396161 (1-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396208 (6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396224 (3-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Homo sapiens (Human)) | BDBM396229 (6-[5-Bromo-6-(3,3-difluoro-pyrrolidin-1-yl)-pyridi...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim Pharmaceuticals Inc. | Assay Description Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,... | Bioorg Med Chem Lett 17: 4664-9 (2007) BindingDB Entry DOI: 10.7270/Q2VH5R5S | |||||||||||
More data for this Ligand-Target Pair |
Displayed 1 to 50 (of 312 total ) | Next | Last >> |