Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218810 (NTS8-13) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM85050 (CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218811 (NTSR-H4 inhibitor, 1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218812 (NTSR-H4 inhibitor, 2) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218813 (NTSR-H4 inhibitor, 3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218815 (NTSR-H4 inhibitor, 5) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.15E+4 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218815 (NTSR-H4 inhibitor, 5) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.20E+4 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218811 (NTSR-H4 inhibitor, 1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218812 (NTSR-H4 inhibitor, 2) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218813 (NTSR-H4 inhibitor, 3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218814 (NTSR-H4 inhibitor, 4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.76E+4 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A] (Rattus norvegicus (Rat)) | BDBM218814 (NTSR-H4 inhibitor, 4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a |
Stockholm University | Assay Description The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused... | ACS Chem Biol 12: 735-745 (2017) Article DOI: 10.1021/acschembio.6b00646 BindingDB Entry DOI: 10.7270/Q2542MFK | |||||||||||
More data for this Ligand-Target Pair |