Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nociceptin receptor (Cavia porcellus) | BDBM50189257 (CHEMBL378753 | NalBzOH) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (GUINEA PIG) | BDBM50000788 ((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Hungarian Academy of Sciences Curated by PDSP Ki Database | Eur J Pharmacol 383: 209-14 (1999) Article DOI: 10.1016/s0014-2999(99)00610-x BindingDB Entry DOI: 10.7270/Q2TT4PJ9 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189252 (CHEMBL214040 | M3A6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 5.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189247 (CHEMBL1418 | M6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189258 (CHEMBL385448 | DM6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189251 (CHEMBL213228 | M3P6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50000092 ((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189256 (CHEMBL385048 | M3Pr6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM21015 ((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189249 (CHEMBL211576 | M3IBu6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 266 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50019056 ((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 277 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189250 (CHEMBL379928 | MM3A6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189259 (C6S | CHEMBL1417) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 455 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189260 (CHEMBL209751 | M3B6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 513 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189245 (CHEMBL1416 | DC6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 760 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189253 (CHEMBL213737 | DM3B6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 822 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189246 (CHEMBL437682 | DM3A6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 838 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50068133 ((4S,7S,13S)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50381677 (CHEMBL1256748 | U-69593) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189254 (CHEMBL1415 | M3S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 1.69E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50189248 (CHEMBL211374 | MM3B6S) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kentucky Curated by ChEMBL | Assay Description Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brain | Bioorg Med Chem Lett 16: 4291-5 (2006) Article DOI: 10.1016/j.bmcl.2006.05.060 BindingDB Entry DOI: 10.7270/Q2XG9RXF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50475333 (CHEMBL264846) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Inhibition of electrically evoked contraction of guinea pig ileum | J Med Chem 48: 1421-7 (2005) Article DOI: 10.1021/jm040106v BindingDB Entry DOI: 10.7270/Q2J38WBW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50411362 (CHEMBL437744) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 0.316 | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Antagonist activity at NOP receptor in Albino guinea pig ileum assessed as effect on electrically stimulated contractions | Bioorg Med Chem 15: 4434-43 (2007) Article DOI: 10.1016/j.bmc.2007.04.026 BindingDB Entry DOI: 10.7270/Q22R3SVP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50475328 (CHEMBL414782) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Inhibition of electrically evoked contraction of guinea pig ileum | J Med Chem 48: 1421-7 (2005) Article DOI: 10.1021/jm040106v BindingDB Entry DOI: 10.7270/Q2J38WBW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50475327 (CHEMBL410653) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Inhibition of electrically evoked contraction of guinea pig ileum | J Med Chem 48: 1421-7 (2005) Article DOI: 10.1021/jm040106v BindingDB Entry DOI: 10.7270/Q2J38WBW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin receptor (Cavia porcellus) | BDBM50004178 (Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Inhibition of electrically evoked contraction of guinea pig ileum | J Med Chem 48: 1421-7 (2005) Article DOI: 10.1021/jm040106v BindingDB Entry DOI: 10.7270/Q2J38WBW | |||||||||||
More data for this Ligand-Target Pair |