Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein kinase C eta type (Mus musculus) | BDBM50064089 (4-hydroxymethyl-7,10-diisopropyl-8,10,13-trimethyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C eta | Bioorg Med Chem Lett 6: 353-356 (1996) Article DOI: 10.1016/0960-894X(96)00026-1 BindingDB Entry DOI: 10.7270/Q2NG4QMM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50057514 ((10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-5...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]- PDBu from Protein kinase C delta C1b domain | J Med Chem 45: 853-60 (2002) BindingDB Entry DOI: 10.7270/Q20C4V25 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50133235 (CHEMBL132720 | Docosanedioic acid ((S)-5-hydroxyme...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [... | J Med Chem 46: 4196-204 (2003) Article DOI: 10.1021/jm0302041 BindingDB Entry DOI: 10.7270/Q2GF0SX2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50099646 (5,6-dihydroxy-7-hydroxymethyl-3,11,11,14-tetrameth...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 0.130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain (Wild type) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50133238 (CHEMBL334853 | Hexadecanedioic acid ((S)-5-hydroxy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [... | J Med Chem 46: 4196-204 (2003) Article DOI: 10.1021/jm0302041 BindingDB Entry DOI: 10.7270/Q2GF0SX2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50099646 (5,6-dihydroxy-7-hydroxymethyl-3,11,11,14-tetrameth...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 0.150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (F13G) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50133236 (CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.330 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [... | J Med Chem 46: 4196-204 (2003) Article DOI: 10.1021/jm0302041 BindingDB Entry DOI: 10.7270/Q2GF0SX2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50057512 ((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 0.330 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute-Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from mouse wild type C1b domain of PKCdelta expressed in Escherichia coli | J Med Chem 50: 3465-81 (2007) Article DOI: 10.1021/jm0702579 BindingDB Entry DOI: 10.7270/Q2RF5TQ5 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50080322 (Acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-9-acet...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.351 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Binding of Indolactam-V(ILV) to wild-type Protein kinase C delta C1b domain | J Med Chem 42: 3436-46 (1999) Article DOI: 10.1021/jm990129n BindingDB Entry DOI: 10.7270/Q25T3JP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50057512 ((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | 0.351 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain (Wild type) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50133238 (CHEMBL334853 | Hexadecanedioic acid ((S)-5-hydroxy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.360 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+] | J Med Chem 46: 4196-204 (2003) Article DOI: 10.1021/jm0302041 BindingDB Entry DOI: 10.7270/Q2GF0SX2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50133235 (CHEMBL132720 | Docosanedioic acid ((S)-5-hydroxyme...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+] | J Med Chem 46: 4196-204 (2003) Article DOI: 10.1021/jm0302041 BindingDB Entry DOI: 10.7270/Q2GF0SX2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50133249 (CHEMBL133853 | Dodecanedioic acid [(S)-5-hydroxyme...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.480 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [... | J Med Chem 46: 4196-204 (2003) Article DOI: 10.1021/jm0302041 BindingDB Entry DOI: 10.7270/Q2GF0SX2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C eta type (Mus musculus) | BDBM50057512 ((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C eta | Bioorg Med Chem Lett 6: 353-356 (1996) Article DOI: 10.1016/0960-894X(96)00026-1 BindingDB Entry DOI: 10.7270/Q2NG4QMM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50099646 (5,6-dihydroxy-7-hydroxymethyl-3,11,11,14-tetrameth...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 0.720 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T12G) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50554605 (CHEMBL4755092) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.740 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of [3H]-PDBu from PKCdelta C1B domain in CD-1 mouse brain cytosol | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127657 BindingDB Entry DOI: 10.7270/Q2SB49DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50133236 (CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.780 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+] | J Med Chem 46: 4196-204 (2003) Article DOI: 10.1021/jm0302041 BindingDB Entry DOI: 10.7270/Q2GF0SX2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50057512 ((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | 0.820 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (F13G) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50216859 (CHEMBL442232 | {2-(hydroxymethyl)-5-[5-methyl-3-(2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.820 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute-Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from mouse wild type C1b domain of PKCdelta expressed in Escherichia coli | J Med Chem 50: 3465-81 (2007) Article DOI: 10.1021/jm0702579 BindingDB Entry DOI: 10.7270/Q2RF5TQ5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50080322 (Acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-9-acet...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.820 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Binding of Indolactam-V(ILV) to mutant Protein kinase C delta C1b domain (Phe13 to Gly) | J Med Chem 42: 3436-46 (1999) Article DOI: 10.1021/jm990129n BindingDB Entry DOI: 10.7270/Q25T3JP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50216857 ((2-(hydroxymethyl)-4-(3-methylbutylidene)-5-oxo-te...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute-Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from mouse wild type C1b domain of PKCdelta expressed in Escherichia coli | J Med Chem 50: 3465-81 (2007) Article DOI: 10.1021/jm0702579 BindingDB Entry DOI: 10.7270/Q2RF5TQ5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50216856 (CHEMBL231617 | Z-{2-(Hydroxymethyl)-4-[5-methyl-3-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.960 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute-Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from mouse wild type C1b domain of PKCdelta expressed in Escherichia coli | J Med Chem 50: 3465-81 (2007) Article DOI: 10.1021/jm0702579 BindingDB Entry DOI: 10.7270/Q2RF5TQ5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50554604 (CHEMBL4763383) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.980 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of [3H]-PDBu from PKCdelta C1B domain in CD-1 mouse brain cytosol | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127657 BindingDB Entry DOI: 10.7270/Q2SB49DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50099646 (5,6-dihydroxy-7-hydroxymethyl-3,11,11,14-tetrameth...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 1.08 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (L20G) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50107112 ((Z) 2,2-Dimethyl-propionic acid 2-hydroxymethyl-4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute-Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from mouse wild type C1b domain of PKCdelta expressed in Escherichia coli | J Med Chem 50: 3465-81 (2007) Article DOI: 10.1021/jm0702579 BindingDB Entry DOI: 10.7270/Q2RF5TQ5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50107112 ((Z) 2,2-Dimethyl-propionic acid 2-hydroxymethyl-4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute-Frederick Curated by ChEMBL | Assay Description Binding affinity to mouse wildtype PKCdelta C1a expressed in Escherichia coli | J Med Chem 50: 3465-81 (2007) Article DOI: 10.1021/jm0702579 BindingDB Entry DOI: 10.7270/Q2RF5TQ5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50057512 ((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | 1.24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T12G) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50080322 (Acetic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-9-acet...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Binding of Indolactam-V(ILV) to mutant Protein kinase C delta C1b domain (Thr12 to Gly) | J Med Chem 42: 3436-46 (1999) Article DOI: 10.1021/jm990129n BindingDB Entry DOI: 10.7270/Q25T3JP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50133249 (CHEMBL133853 | Dodecanedioic acid [(S)-5-hydroxyme...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+] | J Med Chem 46: 4196-204 (2003) Article DOI: 10.1021/jm0302041 BindingDB Entry DOI: 10.7270/Q2GF0SX2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50133243 (CHEMBL132612 | Decanedioic acid ((S)-5-hydroxymeth...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [... | J Med Chem 46: 4196-204 (2003) Article DOI: 10.1021/jm0302041 BindingDB Entry DOI: 10.7270/Q2GF0SX2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50099646 (5,6-dihydroxy-7-hydroxymethyl-3,11,11,14-tetrameth...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 1.41 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (Q27V) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50057511 ((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PubMed | 2.01 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]- PDBu from Protein kinase C delta C1b domain | J Med Chem 45: 853-60 (2002) BindingDB Entry DOI: 10.7270/Q20C4V25 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50057511 ((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 2.01 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Binding of Indolactam-V(ILV) to wild-type Protein kinase C delta C1b domain | J Med Chem 42: 3436-46 (1999) Article DOI: 10.1021/jm990129n BindingDB Entry DOI: 10.7270/Q25T3JP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50057511 ((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PubMed | 2.01 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain (Wild type) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244416 (CHEMBL527875 | rac-(E)-{4-[(3-Bromo-4-fluorophenyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.07 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244416 (CHEMBL527875 | rac-(E)-{4-[(3-Bromo-4-fluorophenyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.07 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50216860 (CHEMBL230048 | Z-[2-(Hydroxymethyl)-4-(3-methylbut...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute-Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from mouse wild type C1b domain of PKCdelta expressed in Escherichia coli | J Med Chem 50: 3465-81 (2007) Article DOI: 10.1021/jm0702579 BindingDB Entry DOI: 10.7270/Q2RF5TQ5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244693 (CHEMBL516638 | rac-(E)-{4-[(3-Chloro-4-fluoropheny...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.45 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244693 (CHEMBL516638 | rac-(E)-{4-[(3-Chloro-4-fluoropheny...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.45 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244961 (CHEMBL472520 | rac-(E/Z)-(4-heptylidene-2-(hydroxy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244961 (CHEMBL472520 | rac-(E/Z)-(4-heptylidene-2-(hydroxy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244413 (CHEMBL488498 | rac-(E)-{4-[(3-Bromo-4-fluorophenyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.66 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244413 (CHEMBL488498 | rac-(E)-{4-[(3-Bromo-4-fluorophenyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.66 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50099645 (CHEMBL49689 | Thymeleatoxin) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 2.71 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Georgetown University Medical Center Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from protein kinase C delta C1b domain (Wild type) | J Med Chem 44: 1690-701 (2001) BindingDB Entry DOI: 10.7270/Q2RR1ZX3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Mus musculus) | BDBM50216858 ((Z)-(2-(hydroxymethyl)-4-(3-isobutyl-5-methylhexyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.82 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute-Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from mouse wild type C1b domain of PKCdelta expressed in Escherichia coli | J Med Chem 50: 3465-81 (2007) Article DOI: 10.1021/jm0702579 BindingDB Entry DOI: 10.7270/Q2RF5TQ5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244414 (CHEMBL488500 | rac-(E)-{4-[(4-Chlorophenyl)methyle...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50107112 ((Z) 2,2-Dimethyl-propionic acid 2-hydroxymethyl-4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute-Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu from mouse recombinant PKCalpha expressed in Escherichia coli | J Med Chem 50: 3465-81 (2007) Article DOI: 10.1021/jm0702579 BindingDB Entry DOI: 10.7270/Q2RF5TQ5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244414 (CHEMBL488500 | rac-(E)-{4-[(4-Chlorophenyl)methyle...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244648 (CHEMBL453598 | rac-(E)-(2-(Hydroxymethyl)-5-oxo-4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.96 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (MOUSE) | BDBM50244648 (CHEMBL453598 | rac-(E)-(2-(Hydroxymethyl)-5-oxo-4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.96 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Cancer Institute at Frederick Curated by ChEMBL | Assay Description Displacement of [3H]PDBu form mouse PKCalpha by scintillation counting | J Med Chem 51: 5198-220 (2008) Article DOI: 10.1021/jm8001907 BindingDB Entry DOI: 10.7270/Q2G44Q4B | |||||||||||
More data for this Ligand-Target Pair |
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