Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50121975 ((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213095 ((1S,2S)-1-(1-Naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50131434 (CHEMBL652 | FLECAINIDE | N-(piperidin-2-ylmethyl)-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213093 ((1R,2R)-1-(1-naphthalenethoxy)-2-(3-ketopyrrolidin...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213094 ((1R,2R)-1-(3,4-dichlorophenethoxy)-2-(4-morpholiny...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50213092 ((1R,2R)-1-(1-naphthalenethoxy)-2-(4-morpholinyl)cy...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily D member 2 (Rattus norvegicus) | BDBM50017662 (2-(Diethylamino)-2',6'-acetoxylidide | 2-(Diethyla...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.21E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiome Pharma Corporation Curated by ChEMBL | Assay Description Inhibition of rat potassium channel Kv4.2 by patch-clamp method | J Med Chem 50: 2818-41 (2007) Article DOI: 10.1021/jm0604528 BindingDB Entry DOI: 10.7270/Q29Z95QZ | |||||||||||
More data for this Ligand-Target Pair |