Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Xanthine-guanine phosphoribosyltransferase (Escherichia coli (strain K12)) | BDBM194503 (US9200020, 1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 400 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
THE UNIVERSITY OF QUEENSLAND; INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY ASCR, V.V.I. US Patent | Assay Description The Ki values were determined using a spectrophotometric assay at 25° C., 0.1 M Tris-HCl, 10 mM MgCl2, pH 7.4 (Keough, D. T.; Ng, A. L.; Winzor, D. J... | US Patent US9200020 (2015) BindingDB Entry DOI: 10.7270/Q2TM78XB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Xanthine-guanine phosphoribosyltransferase (Escherichia coli (strain K12)) | BDBM194504 (US9200020, 2) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 2.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
THE UNIVERSITY OF QUEENSLAND; INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY ASCR, V.V.I. US Patent | Assay Description The Ki values were determined using a spectrophotometric assay at 25° C., 0.1 M Tris-HCl, 10 mM MgCl2, pH 7.4 (Keough, D. T.; Ng, A. L.; Winzor, D. J... | US Patent US9200020 (2015) BindingDB Entry DOI: 10.7270/Q2TM78XB | |||||||||||
More data for this Ligand-Target Pair |