Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179292 (US9125915, compound 17) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 12.8 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179288 (US9125915, compound 13) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 17.3 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179283 (US9125915, compound 6) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | PDB US Patent | n/a | n/a | 18.2 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179289 (US9125915, compound 14) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179277 (US9125915, compound 10) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 47.1 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179282 (US9125915, compound 5) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 54.2 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179280 (US9125915, compound 3) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 54.9 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179285 (US9125915, compound 9) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 73.6 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179281 (US9125915, compound 4) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 77.2 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179287 (US9125915, compound 12) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 108 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179276 (US9125915, compound 7) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 113 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179291 (US9125915, compound 16) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 116 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179290 (US9125915, compound 15) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179275 (US9125915, compound 2) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 121 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179284 (US9125915, compound 8) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 124 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179279 (US9125915, compound 18) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 147 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4/Histone H4 (Homo sapiens (Human)) | BDBM179286 (US9125915, compound 11) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 225 | n/a | n/a | n/a | n/a | n/a | 25 |
Mitsubishi Tanabe Pharma Corporation US Patent | Assay Description An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi... | US Patent US9125915 (2015) BindingDB Entry DOI: 10.7270/Q26972BJ | |||||||||||
More data for this Ligand-Target Pair |