Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Regulator of G-protein signaling 7 (Homo sapiens (Human)) | BDBM34340 (2-(4-methyl-3-piperidin-1-ylsulfonyl-phenyl)-1,2-b...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 140 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2PV6HS7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 19 (Homo sapiens (Human)) | BDBM34340 (2-(4-methyl-3-piperidin-1-ylsulfonyl-phenyl)-1,2-b...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 610 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2K35S27 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 16 (Homo sapiens (Human)) | BDBM34340 (2-(4-methyl-3-piperidin-1-ylsulfonyl-phenyl)-1,2-b...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2FB51BW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 8 (Homo sapiens (Human)) | BDBM34340 (2-(4-methyl-3-piperidin-1-ylsulfonyl-phenyl)-1,2-b...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2TM78JD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Large T antigen (Simian virus 40) | BDBM34340 (2-(4-methyl-3-piperidin-1-ylsulfonyl-phenyl)-1,2-b...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 1.47E+4 | n/a | n/a | n/a | n/a |
Southern Research Specialized Biocontainment Screening Center Curated by PubChem BioAssay | Assay Description Southern Research's Specialized Biocontainment Screening Center (SRSBSC) Southern Research Institute (Birmingham, Alabama) NIH Molecular Librarie... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2ZK5F47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 4 (Homo sapiens (Human)) | BDBM34340 (2-(4-methyl-3-piperidin-1-ylsulfonyl-phenyl)-1,2-b...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2F76B0G | |||||||||||
More data for this Ligand-Target Pair |