Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gastrin-releasing peptide receptor (Homo sapiens (Human)) | BDBM50071745 (CHEMBL403317 | Compound NMB | Gly-Asn-Leu-Trp-Ala-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 41 | n/a | n/a | n/a | n/a |
Technische Universität München Curated by ChEMBL | Assay Description Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assay | J Med Chem 46: 1918-30 (2003) Article DOI: 10.1021/jm0210921 BindingDB Entry DOI: 10.7270/Q29S1QDS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-B receptor (Homo sapiens (Human)) | BDBM50071745 (CHEMBL403317 | Compound NMB | Gly-Asn-Leu-Trp-Ala-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 120 | n/a | n/a | n/a | n/a |
Technische Universität München Curated by ChEMBL | Assay Description Effective concentration required against nueromedin B receptor (NMB-R) in CHO cells by using FLIPR assay | J Med Chem 46: 1918-30 (2003) Article DOI: 10.1021/jm0210921 BindingDB Entry DOI: 10.7270/Q29S1QDS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Homo sapiens (Human)) | BDBM50071745 (CHEMBL403317 | Compound NMB | Gly-Asn-Leu-Trp-Ala-...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.50E+3 | n/a | n/a | n/a | n/a |
Technische Universität München Curated by ChEMBL | Assay Description Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay. | J Med Chem 46: 1918-30 (2003) Article DOI: 10.1021/jm0210921 BindingDB Entry DOI: 10.7270/Q29S1QDS | |||||||||||
More data for this Ligand-Target Pair |