Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucagon-like peptide 1 receptor (Homo sapiens (Human)) | BDBM50086603 (CHEMBL3426241) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.120 | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Agonist activity at human GLP-1R expressed in CHO cells assessed as cAMP accumulation incubated for 30 mins | J Med Chem 58: 4080-5 (2015) Article DOI: 10.1021/acs.jmedchem.5b00166 BindingDB Entry DOI: 10.7270/Q2DB83KP | |||||||||||
More data for this Ligand-Target Pair |