Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Retinoic acid receptor RXR-alpha (Homo sapiens (Human)) | BDBM50101446 ((2E,4E)-3-Methyl-5-[(1R,2R)-2-methyl-2-(5,5,8,8-te...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Allergan Inc. Curated by ChEMBL | Assay Description Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alpha | J Med Chem 44: 2298-303 (2001) BindingDB Entry DOI: 10.7270/Q2P84B41 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor RXR-gamma (Homo sapiens (Human)) | BDBM50101446 ((2E,4E)-3-Methyl-5-[(1R,2R)-2-methyl-2-(5,5,8,8-te...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Allergan Inc. Curated by ChEMBL | Assay Description Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gamma | J Med Chem 44: 2298-303 (2001) BindingDB Entry DOI: 10.7270/Q2P84B41 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor RXR-beta (Homo sapiens (Human)) | BDBM50101446 ((2E,4E)-3-Methyl-5-[(1R,2R)-2-methyl-2-(5,5,8,8-te...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
Allergan Inc. Curated by ChEMBL | Assay Description Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR beta | J Med Chem 44: 2298-303 (2001) BindingDB Entry DOI: 10.7270/Q2P84B41 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50101446 ((2E,4E)-3-Methyl-5-[(1R,2R)-2-methyl-2-(5,5,8,8-te...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | >500 | n/a | n/a | n/a | n/a |
Allergan Inc. Curated by ChEMBL | Assay Description Transcriptional activation in CV-1 cells expressing retinoic acid receptor RAR gamma | J Med Chem 44: 2298-303 (2001) BindingDB Entry DOI: 10.7270/Q2P84B41 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor beta (Homo sapiens (Human)) | BDBM50101446 ((2E,4E)-3-Methyl-5-[(1R,2R)-2-methyl-2-(5,5,8,8-te...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | >500 | n/a | n/a | n/a | n/a |
Allergan Inc. Curated by ChEMBL | Assay Description Transcriptional activation in CV-1 cells expressing retinoic acid receptor RAR beta | J Med Chem 44: 2298-303 (2001) BindingDB Entry DOI: 10.7270/Q2P84B41 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50101446 ((2E,4E)-3-Methyl-5-[(1R,2R)-2-methyl-2-(5,5,8,8-te...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | >500 | n/a | n/a | n/a | n/a |
Allergan Inc. Curated by ChEMBL | Assay Description Transcriptional activation in CV-1 cells expressing retinoic acid receptor RAR alpha | J Med Chem 44: 2298-303 (2001) BindingDB Entry DOI: 10.7270/Q2P84B41 | |||||||||||
More data for this Ligand-Target Pair |