Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha (Mus musculus) | BDBM50126320 (1-{[(4-Cyano-phenyl)-(3-methyl-3H-imidazol-4-yl)-m...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro inhibition of geranylgeranyltransferase-1 | Bioorg Med Chem Lett 13: 1363-6 (2003) BindingDB Entry DOI: 10.7270/Q24B30PD | |||||||||||
More data for this Ligand-Target Pair |