Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Homo sapiens (Human)) | BDBM50229056 (CHEMBL349025) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | n/a | n/a | 150 | n/a | n/a | n/a | n/a |
Ferrosan A/S Curated by ChEMBL | Assay Description Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum. | J Med Chem 34: 687-92 (1991) BindingDB Entry DOI: 10.7270/Q2RN3B25 | |||||||||||
More data for this Ligand-Target Pair |