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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50356038   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucocorticoid receptor


(Homo sapiens (Human))		BDBM50356038
PNG
(CHEMBL1911544)
Show SMILES COc1ccc(F)cc1C(C)(C)CC(O)(Cc1cc2cccc(F)c2[nH]1)C(F)(F)F
Show InChI InChI=1S/C22H22F5NO2/c1-20(2,16-10-14(23)7-8-18(16)30-3)12-21(29,22(25,26)27)11-15-9-13-5-4-6-17(24)19(13)28-15/h4-10,28-29H,11-12H2,1-3H3
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Article
PubMed
n/an/an/an/a 473n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL


Assay Description
Transactivation activity of glucocorticoid receptor in HFF assessed as induction of aromatase activity by measuring beta-estradiol activity after 18 ...

Bioorg Med Chem Lett 21: 6842-51 (2011)


Article DOI: 10.1016/j.bmcl.2011.09.018
BindingDB Entry DOI: 10.7270/Q2CV4J51
More data for this
Ligand-Target Pair