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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50388683   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Muscarinic acetylcholine receptor M1


(Homo sapiens (Human))		BDBM50388683
PNG
(CHEMBL2059322)
Show SMILES Fc1ccc2[nH]c(=O)n(C3CCN(CCCN4C(=O)COc5ccccc45)CC3)c2c1
Show InChI InChI=1S/C23H25FN4O3/c24-16-6-7-18-20(14-16)28(23(30)25-18)17-8-12-26(13-9-17)10-3-11-27-19-4-1-2-5-21(19)31-15-22(27)29/h1-2,4-7,14,17H,3,8-13,15H2,(H,25,30)
UniProtKB/SwissProt

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PC sid
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Similars
Article
PubMed
n/an/an/an/a 44n/an/an/an/a



H. Lundbeck A/S

Curated by ChEMBL


Assay Description
Agonist activity at human M1 receptor expressed in CHO-K1 cells assessed as calcium mobilization for 6 mins by Calcium4-based staining

Bioorg Med Chem Lett 22: 5134-40 (2012)


Article DOI: 10.1016/j.bmcl.2012.05.048
BindingDB Entry DOI: 10.7270/Q24M95MM
More data for this
Ligand-Target Pair