Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50392401 (CHEMBL2151642) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0650 | n/a | n/a | n/a | n/a |
Takeda Pharmaceutical Company Ltd Curated by ChEMBL | Assay Description Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysis | Bioorg Med Chem Lett 22: 6391-6 (2012) Article DOI: 10.1016/j.bmcl.2012.08.069 BindingDB Entry DOI: 10.7270/Q2ZP477R | |||||||||||
More data for this Ligand-Target Pair |