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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50432157   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Extracellular calcium-sensing receptor


(Homo sapiens (Human))		BDBM50432157
PNG
(CHEMBL2346778)
Show SMILES OC(=O)c1cccc(NC(=O)NCCC(c2ccccc2)c2ccccc2)c1
Show InChI InChI=1S/C23H22N2O3/c26-22(27)19-12-7-13-20(16-19)25-23(28)24-15-14-21(17-8-3-1-4-9-17)18-10-5-2-6-11-18/h1-13,16,21H,14-15H2,(H,26,27)(H2,24,25,28)
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Article
PubMed
n/an/an/an/a 2.00E+4n/an/an/an/a



Galapagos SASU

Curated by ChEMBL


Assay Description
Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assay

Bioorg Med Chem Lett 23: 2451-4 (2013)


Article DOI: 10.1016/j.bmcl.2013.01.078
BindingDB Entry DOI: 10.7270/Q2930VJZ
More data for this
Ligand-Target Pair