Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (GUINEA PIG) | BDBM22911 (2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide |...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article | n/a | n/a | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Histamine H3 receptor agonist activity was assessed by the inhibition of the electrically evoked twitch response of the guinea-pig ileum. | Bioorg Med Chem Lett 2: 77-78 (1992) Article DOI: 10.1016/S0960-894X(00)80659-9 BindingDB Entry DOI: 10.7270/Q2222TN4 | |||||||||||
More data for this Ligand-Target Pair |