Compile Data Set for Download or QSAR

Found 2 hits of ic50 for monomerid = 2586   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
cAMP-dependent protein kinase catalytic subunit alpha (Bos taurus (bovine))	BDBM2586 (3,4-Bis(3-indolyl)-3-pyrrolin-2-one | 3,4-bis(1H-i...) Show SMILES O=C1NCC(=C1c1c[nH]c2ccccc12)c1c[nH]c2ccccc12 |c:4| Show InChI InChI=1S/C20H15N3O/c24-20-19(15-10-22-18-8-4-2-6-13(15)18)16(11-23-20)14-9-21-17-7-3-1-5-12(14)17/h1-10,21-22H,11H2,(H,23,24)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a	7.4	30
Laboratoires Glaxo					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Biol Chem 266: 15771-81 (1991) BindingDB Entry DOI: 10.7270/Q2FF3QJ4
					More data for this Ligand-Target Pair
Protein kinase C beta type (Rattus norvegicus (rat))	BDBM2586 (3,4-Bis(3-indolyl)-3-pyrrolin-2-one | 3,4-bis(1H-i...) Show SMILES O=C1NCC(=C1c1c[nH]c2ccccc12)c1c[nH]c2ccccc12 |c:4| Show InChI InChI=1S/C20H15N3O/c24-20-19(15-10-22-18-8-4-2-6-13(15)18)16(11-23-20)14-9-21-17-7-3-1-5-12(14)17/h1-10,21-22H,11H2,(H,23,24)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1.03E+4	n/a	n/a	n/a	n/a	7.5	30
Roche Products Limited					Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...				J Med Chem 35: 177-84 (1992) Article DOI: 10.1021/jm00079a024 BindingDB Entry DOI: 10.7270/Q2K64G8V
					More data for this Ligand-Target Pair