Compile Data Set for Download or QSAR

Found 4 hits of ic50 for monomerid = 276039   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Lysine-specific demethylase 2B (Homo sapiens (Human))	BDBM276039 (2-(1-methylimidazol-4-yl)-4-(1H-triazol-4-yl)pyrid...) Show SMILES Cn1cnc(c1)-c1cc(ccn1)-c1c[nH]nn1 Show InChI InChI=1S/C11H10N6/c1-17-6-11(13-7-17)9-4-8(2-3-12-9)10-5-14-16-15-10/h2-7H,1H3,(H,14,15,16)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	300	n/a	n/a	n/a	n/a	n/a	n/a
GSK					Assay Description The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...				Bioorg Med Chem Lett 17: 1584-9 (2007) BindingDB Entry DOI: 10.7270/Q2FT8PBQ
					More data for this Ligand-Target Pair
Histone lysine demethylase PHF8 (Homo sapiens (Human))	BDBM276039 (2-(1-methylimidazol-4-yl)-4-(1H-triazol-4-yl)pyrid...) Show SMILES Cn1cnc(c1)-c1cc(ccn1)-c1c[nH]nn1 Show InChI InChI=1S/C11H10N6/c1-17-6-11(13-7-17)9-4-8(2-3-12-9)10-5-14-16-15-10/h2-7H,1H3,(H,14,15,16)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	300	n/a	n/a	n/a	n/a	n/a	n/a
GSK					Assay Description PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...				Bioorg Med Chem Lett 17: 1584-9 (2007) BindingDB Entry DOI: 10.7270/Q2FT8PBQ
					More data for this Ligand-Target Pair
Lysine-specific demethylase 2B (Homo sapiens (Human))	BDBM276039 (2-(1-methylimidazol-4-yl)-4-(1H-triazol-4-yl)pyrid...) Show SMILES Cn1cnc(c1)-c1cc(ccn1)-c1c[nH]nn1 Show InChI InChI=1S/C11H10N6/c1-17-6-11(13-7-17)9-4-8(2-3-12-9)10-5-14-16-15-10/h2-7H,1H3,(H,14,15,16)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10071984 (2018) BindingDB Entry DOI: 10.7270/Q24Q7X0X
					More data for this Ligand-Target Pair
Isoform 2 of Histone lysine demethylase PHF8 (2) (Homo sapiens (Human))	BDBM276039 (2-(1-methylimidazol-4-yl)-4-(1H-triazol-4-yl)pyrid...) Show SMILES Cn1cnc(c1)-c1cc(ccn1)-c1c[nH]nn1 Show InChI InChI=1S/C11H10N6/c1-17-6-11(13-7-17)9-4-8(2-3-12-9)10-5-14-16-15-10/h2-7H,1H3,(H,14,15,16)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction conditions: 3 nM P...				US Patent US10071984 (2018) BindingDB Entry DOI: 10.7270/Q24Q7X0X
					More data for this Ligand-Target Pair