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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50018315   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50018315
PNG
(2-Ethynyl-3',4'-dimethoxy-biphenyl-4-carboxylic ac...)
Show SMILES COc1ccc(cc1OC)-c1ccc(cc1C#C)C(=O)N[C@H](C)CCCc1cccnc1
Show InChI InChI=1S/C27H28N2O3/c1-5-21-16-23(11-13-24(21)22-12-14-25(31-3)26(17-22)32-4)27(30)29-19(2)8-6-9-20-10-7-15-28-18-20/h1,7,10-19H,6,8-9H2,2-4H3,(H,29,30)/t19-/m1/s1
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Roche Research Center

Curated by ChEMBL


Assay Description
Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.

J Med Chem 32: 1814-20 (1989)


BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ
More data for this
Ligand-Target Pair