Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 1 (RAT) | BDBM50034503 ((1R,2R)-3-((S)-Amino-carboxy-methyl)-cyclopropane-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 3.89E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Parc Club Orsay Université Curated by ChEMBL | Assay Description Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells. | J Med Chem 42: 1546-55 (1999) Article DOI: 10.1021/jm980571q BindingDB Entry DOI: 10.7270/Q27H1HRD | |||||||||||
More data for this Ligand-Target Pair |