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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50090426   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Protein c-Fos/Transcription factor Jun


(Homo sapiens (Human))		BDBM50090426
PNG
(2-(4-Fluoro-phenyl)-4-(3-methyl-2,5-dioxo-2,5-dihy...)
Show SMILES CCOC(=O)c1cnc(nc1NN1C(=O)C=C(C)C1=O)-c1ccc(F)cc1 |t:16|
Show InChI InChI=1S/C18H15FN4O4/c1-3-27-18(26)13-9-20-15(11-4-6-12(19)7-5-11)21-16(13)22-23-14(24)8-10(2)17(23)25/h4-9H,3H2,1-2H3,(H,20,21,22)
PDB

KEGG

UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem

Similars
PubMed
n/an/a 700n/an/an/an/an/an/a



Signal Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cells

Bioorg Med Chem Lett 10: 1645-8 (2000)


BindingDB Entry DOI: 10.7270/Q2F190XH
More data for this
Ligand-Target Pair