Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
LIM domain kinase 1 (Homo sapiens (Human)) | BDBM50130039 (CHEMBL3629276) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Institute of Technology Curated by ChEMBL | Assay Description Inhibition of LIMK1 (unknown origin) using 1 uM cofilin as substrate | Bioorg Med Chem 23: 7464-77 (2015) Article DOI: 10.1016/j.bmc.2015.10.041 BindingDB Entry DOI: 10.7270/Q2Q81FW9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 2 (Homo sapiens (Human)) | BDBM50130039 (CHEMBL3629276) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Institute of Technology Curated by ChEMBL | Assay Description Inhibition of ROCK2 (unknown origin) after 4 hrs using 1 uM STK2 as substrate | Bioorg Med Chem 23: 7464-77 (2015) Article DOI: 10.1016/j.bmc.2015.10.041 BindingDB Entry DOI: 10.7270/Q2Q81FW9 | |||||||||||
More data for this Ligand-Target Pair |