Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tubulin alpha-1A chain (Sus scrofa (Pig)) | BDBM50134461 (2-(3-Hydroxy-4-methoxy-phenyl)-5,6,7-trimethoxy-ch...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiff University Curated by ChEMBL | Assay Description Concentration that cause a 50% inhibition in tubulin assembly as measured by an increase inturbidity using microtubule assembly assay | Bioorg Med Chem Lett 13: 3759-63 (2003) BindingDB Entry DOI: 10.7270/Q2G73D48 | |||||||||||
More data for this Ligand-Target Pair |