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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50213748   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
C-X-C chemokine receptor type 2


(Homo sapiens (Human))		BDBM50213748
PNG
(7-chloro-3-(2-morpholin-4-yl-phenylamino)-1,1-diox...)
Show SMILES Oc1cc(Cl)cc2c1N=C(Nc1ccccc1N1CCOCC1)NS2(=O)=O |t:9|
Show InChI InChI=1S/C17H17ClN4O4S/c18-11-9-14(23)16-15(10-11)27(24,25)21-17(20-16)19-12-3-1-2-4-13(12)22-5-7-26-8-6-22/h1-4,9-10,23H,5-8H2,(H2,19,20,21)
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PC cid
PC sid
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Article
PubMed
n/an/a>3.00E+4n/an/an/an/an/an/a



GlaxoSmithKline

Curated by ChEMBL


Assay Description
Antagonist activity at CXCR2 receptor expressed in CHOK1 cells assessed as human IL8-induced calcium mobilization by FLIPR

Bioorg Med Chem Lett 17: 3864-7 (2007)


Article DOI: 10.1016/j.bmcl.2007.05.011
BindingDB Entry DOI: 10.7270/Q21C1WKG
More data for this
Ligand-Target Pair