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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50301087   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50301087
PNG
(4-(4-fluorobenzyloxy)-1-(4-(pyrrolidin-1-yl)phenet...)
Show SMILES Fc1ccc(COc2ccn(CCc3ccc(cc3)N3CCCC3)c(=O)c2)cc1
Show InChI InChI=1S/C24H25FN2O2/c25-21-7-3-20(4-8-21)18-29-23-12-16-27(24(28)17-23)15-11-19-5-9-22(10-6-19)26-13-1-2-14-26/h3-10,12,16-17H,1-2,11,13-15,18H2
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PC cid
PC sid
UniChem
Article
PubMed
n/an/a>1.00E+3n/an/an/an/an/an/a



Tsukuba Research Institute

Curated by ChEMBL


Assay Description
Antagonistic activity against MCH1R expressed on CHOK1 cells assessed as intracellular calcium mobilization by FLIPR

Bioorg Med Chem Lett 19: 5186-90 (2009)


Article DOI: 10.1016/j.bmcl.2009.07.023
BindingDB Entry DOI: 10.7270/Q2G44QCG
More data for this
Ligand-Target Pair