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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50312583   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Cannabinoid receptor 1


(Homo sapiens (Human))		BDBM50312583
PNG
(CHEMBL1087875 | N-cyclohexyl-4-((3,4-dichloropheny...)
Show SMILES Clc1ccc(cc1Cl)C(N1CCN(CC1)C(=O)NC1CCCCC1)c1ccccc1
Show InChI InChI=1S/C24H29Cl2N3O/c25-21-12-11-19(17-22(21)26)23(18-7-3-1-4-8-18)28-13-15-29(16-14-28)24(30)27-20-9-5-2-6-10-20/h1,3-4,7-8,11-12,17,20,23H,2,5-6,9-10,13-16H2,(H,27,30)
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Similars
Article
PubMed
n/an/a 462n/an/an/an/an/an/a



Chinese Academy of Sciences

Curated by ChEMBL


Assay Description
Antagonist activity at human cannabinoid CB1 receptor expressed in CHO cells coexpressing Galpha15/16 assessed as inhibition of CP55940-induced Ca2+ ...

Eur J Med Chem 45: 1133-9 (2010)


Article DOI: 10.1016/j.ejmech.2009.12.018
BindingDB Entry DOI: 10.7270/Q2K937P0
More data for this
Ligand-Target Pair