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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50448087   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Phosphatidylinositol 4-kinase alpha


(Homo sapiens (Human))		BDBM50448087
PNG
(CHEMBL3121321)
Show SMILES COc1ncc(cc1NS(=O)(=O)c1ccc(C)cc1)-c1ccc2nc(N)n(-c3ccccc3)c(=O)c2c1
Show InChI InChI=1S/C27H23N5O4S/c1-17-8-11-21(12-9-17)37(34,35)31-24-15-19(16-29-25(24)36-2)18-10-13-23-22(14-18)26(33)32(27(28)30-23)20-6-4-3-5-7-20/h3-16,31H,1-2H3,(H2,28,30)
PDB

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PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/a 16n/an/an/an/an/an/a



GlaxoSmithKline

Curated by ChEMBL


Assay Description
Inhibition of GST-tagged PI4K-alpha (1 to 2044) (unknown origin) using D-myo-phosphatidylinositol as substrate preincubated for 30 mins followed by s...

J Med Chem 57: 2091-106 (2014)


Article DOI: 10.1021/jm400781h
BindingDB Entry DOI: 10.7270/Q2WH2RG0
More data for this
Ligand-Target Pair