Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Casein kinase I isoform alpha (Homo sapiens (Human)) | BDBM92673 (Isoquinolinesulfonamide, CKI-6) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Nagoya University School of Medicine | Assay Description Casein kinase activities were determined under the conditions as described by Huang et al (1982). | J Biol Chem 264: 4924-7 (1989) BindingDB Entry DOI: 10.7270/Q2K072VK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Casein kinase II subunit alpha (Homo sapiens (Human)) | BDBM92673 (Isoquinolinesulfonamide, CKI-6) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Nagoya University School of Medicine | Assay Description Casein kinase activities were determined under the conditions as described by Huang et al (1982). | J Biol Chem 264: 4924-7 (1989) BindingDB Entry DOI: 10.7270/Q2K072VK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcium/calmodulin-dependent protein kinase II inhibitor 2 (Bos taurus (Bovine)) | BDBM92673 (Isoquinolinesulfonamide, CKI-6) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.40E+5 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Nagoya University School of Medicine | Assay Description Casein kinase activities were determined under the conditions as described by Huang et al (1982). | J Biol Chem 264: 4924-7 (1989) BindingDB Entry DOI: 10.7270/Q2K072VK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-dependent protein kinase type I-alpha regulatory subunit (Bos taurus) | BDBM92673 (Isoquinolinesulfonamide, CKI-6) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Nagoya University School of Medicine | Assay Description Casein kinase activities were determined under the conditions as described by Huang et al (1982). | J Biol Chem 264: 4924-7 (1989) BindingDB Entry DOI: 10.7270/Q2K072VK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Homo sapiens (Human)) | BDBM92673 (Isoquinolinesulfonamide, CKI-6) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Nagoya University School of Medicine | Assay Description Casein kinase activities were determined under the conditions as described by Huang et al (1982). | J Biol Chem 264: 4924-7 (1989) BindingDB Entry DOI: 10.7270/Q2K072VK | |||||||||||
More data for this Ligand-Target Pair |