Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM36351 (CID148124 | Docetaxel) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | 0.820 | n/a | n/a | n/a | n/a | n/a |
Veterans Affairs Medical Center Curated by ChEMBL | Assay Description Displacement of radiolabeled EGF from EGF receptor expressed in human MX1 cells | Proc Natl Acad Sci USA 104: 1943-6 (2007) Article DOI: 10.1073/pnas.0610860104 BindingDB Entry DOI: 10.7270/Q28916RX | |||||||||||
More data for this Ligand-Target Pair |