Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Fibroblast growth factor receptor 1 (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 3.10 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor receptor 3 (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 5.40 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor receptor 2 (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mitogen-activated protein kinase 7 (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mast/stem cell growth factor receptor Kit (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor receptor 4 (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vascular endothelial growth factor receptor 3 (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 470 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-derived growth factor receptor beta (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 480 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hepatocyte growth factor receptor (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase Blk (Homo sapiens (Human)) | BDBM81378 (FRIN-1) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a |
Harvard Medical School | Assay Description In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det... | Chem Biol 17: 285-95 (2010) Article DOI: 10.1016/j.chembiol.2010.02.007 BindingDB Entry DOI: 10.7270/Q24B2ZSZ | |||||||||||
More data for this Ligand-Target Pair |