Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50023188 (CHEMBL3298750) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.141 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Catania Curated by ChEMBL | Assay Description Displacement of [125I]BE2254 from human alpha1d receptor expressed in HEK293 cells | Eur J Med Chem 83: 419-32 (2014) Article DOI: 10.1016/j.ejmech.2014.06.057 BindingDB Entry DOI: 10.7270/Q2639RBH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50023188 (CHEMBL3298750) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.324 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Catania Curated by ChEMBL | Assay Description Displacement of [125I]BE2254 from human alpha1a receptor expressed in HEK293 cells | Eur J Med Chem 83: 419-32 (2014) Article DOI: 10.1016/j.ejmech.2014.06.057 BindingDB Entry DOI: 10.7270/Q2639RBH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50023188 (CHEMBL3298750) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.832 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Catania Curated by ChEMBL | Assay Description Displacement of [125I]BE2254 from human alpha1b receptor expressed in HEK293 cells | Eur J Med Chem 83: 419-32 (2014) Article DOI: 10.1016/j.ejmech.2014.06.057 BindingDB Entry DOI: 10.7270/Q2639RBH | |||||||||||
More data for this Ligand-Target Pair |