Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50046128 (2-[2-(2-{2-[2-{2-[3-Carboxy-2-(2-methylamino-3-phe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 0.130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Displacement of [3H]pCCK-8 from cholecystokinin type B receptor in guinea pig brain membrane | J Med Chem 36: 166-72 (1993) BindingDB Entry DOI: 10.7270/Q26M37FJ | |||||||||||
More data for this Ligand-Target Pair |