BindingDB PrimarySearch

Found 5 hits of ki for monomerid = 50236053
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Interleukin-8 receptors, CXCR2 (Homo sapiens (Human))	BDBM50236053 ((R)-3-(3,4-dioxo-2-(1-phenylpropylamino)cyclobut-1...) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents	Article PubMed	4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Schering-Plough Research Institute Curated by ChEMBL					Assay Description Binding affinity to CXCR2 (unknown origin)				Bioorg Med Chem Lett 19: 1431-3 (2009) Article DOI: 10.1016/j.bmcl.2009.01.033 BindingDB Entry DOI: 10.7270/Q2CV4HMF
Schering-Plough Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Interleukin-8 receptors, CXCR2 (Homo sapiens (Human))	BDBM50236053 ((R)-3-(3,4-dioxo-2-(1-phenylpropylamino)cyclobut-1...) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents	Article PubMed	4.40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Schering-Plough Research Institute Curated by ChEMBL					Assay Description Displacement of human [125I]IL-8 from human CXCR2				Bioorg Med Chem Lett 19: 4446-9 (2009) Article DOI: 10.1016/j.bmcl.2009.05.049 BindingDB Entry DOI: 10.7270/Q2H1323X
Schering-Plough Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Interleukin-8 receptors, CXCR2 (Homo sapiens (Human))	BDBM50236053 ((R)-3-(3,4-dioxo-2-(1-phenylpropylamino)cyclobut-1...) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents	Article PubMed	4.70	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Pharmacopeia, Inc. Curated by ChEMBL					Assay Description Displacement of [125I]IL8 from human CXCR2 by SPA assay				Bioorg Med Chem Lett 18: 1864-8 (2008) Article DOI: 10.1016/j.bmcl.2008.02.010 BindingDB Entry DOI: 10.7270/Q2CC10DK
Pharmacopeia, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Chemokine receptor type 1 (CXCR1) (Homo sapiens (Human))	BDBM50236053 ((R)-3-(3,4-dioxo-2-(1-phenylpropylamino)cyclobut-1...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents	Article PubMed	40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Schering-Plough Research Institute Curated by ChEMBL					Assay Description Displacement of human [125I]IL-8 from human CXCR1				Bioorg Med Chem Lett 19: 4446-9 (2009) Article DOI: 10.1016/j.bmcl.2009.05.049 BindingDB Entry DOI: 10.7270/Q2H1323X
Schering-Plough Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Chemokine receptor type 1 (CXCR1) (Homo sapiens (Human))	BDBM50236053 ((R)-3-(3,4-dioxo-2-(1-phenylpropylamino)cyclobut-1...) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents	Article PubMed	40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Schering-Plough Research Institute Curated by ChEMBL					Assay Description Binding affinity to CXCR1 (unknown origin)				Bioorg Med Chem Lett 19: 1431-3 (2009) Article DOI: 10.1016/j.bmcl.2009.01.033 BindingDB Entry DOI: 10.7270/Q2CV4HMF
Schering-Plough Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair