Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Calcitonin gene-related peptide type 1 receptor (Homo sapiens (Human)) | BDBM50301969 (2a-(aminomethyl)-1-(((S)-2'-oxo-1',2',6,8-tetrahyd...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Displacement of [125I]hCGRP from human cloned CGRP receptor expressed in HEK293 cells | Bioorg Med Chem Lett 19: 5787-90 (2009) Article DOI: 10.1016/j.bmcl.2009.07.134 BindingDB Entry DOI: 10.7270/Q2PG1RTW | |||||||||||
More data for this Ligand-Target Pair |