Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Acetylcholinesterase (Electrophorus electricus (Electric eel)) | BDBM50446576 (CHEMBL3109481) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Troms£ Curated by ChEMBL | Assay Description Noncompetitive inhibition of electric eel AChE using acetylthiocholine chloride as substrate after 5 mins by Dixon plot analysis | J Nat Prod 77: 364-9 (2014) Article DOI: 10.1021/np401002s BindingDB Entry DOI: 10.7270/Q2R49S8B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholinesterase (Electrophorus electricus (Electric eel)) | BDBM50446576 (CHEMBL3109481) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Troms£ Curated by ChEMBL | Assay Description Inhibition of electric eel AChE using acetylthiocholine chloride as substrate after 5 mins by Ellman's method | J Nat Prod 77: 364-9 (2014) Article DOI: 10.1021/np401002s BindingDB Entry DOI: 10.7270/Q2R49S8B | |||||||||||
More data for this Ligand-Target Pair |