Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50091725 ((S)-4-(3,4-Difluoro-phenyl)-6-methoxymethyl-2-oxo-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]HEAT from human Alpha-1A adrenergic receptor stably expressed in CHO cells | Bioorg Med Chem Lett 10: 1917-20 (2001) BindingDB Entry DOI: 10.7270/Q2KH0NWK | |||||||||||
More data for this Ligand-Target Pair |