Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50416854 (CHEMBL1254582) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.178 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Bari Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human adrenergic Alpha-1D expressed in CHO cells | Bioorg Med Chem 18: 7065-77 (2010) Article DOI: 10.1016/j.bmc.2010.08.002 BindingDB Entry DOI: 10.7270/Q2B27WKF | |||||||||||
More data for this Ligand-Target Pair |