Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50250521 ((-)-dibromophakellin | CHEMBL447696 | dibromophake...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.20E+3 | n/a | n/a | n/a | n/a |
Griffith University Curated by ChEMBL | Assay Description Agonist activity at human adrenergic alpha2B receptor expressed in HEK293 cells coexpressing Gqi5 protein by FLIPR assay | Bioorg Med Chem 17: 2497-500 (2009) Article DOI: 10.1016/j.bmc.2009.01.065 BindingDB Entry DOI: 10.7270/Q2FJ2GPP | |||||||||||
More data for this Ligand-Target Pair |