Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50320446 (CHEMBL1085510 | [N-methyl]5-methyl-3-[4-(3-phenyla...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by ChEMBL | Assay Description Displacement of [3H]rauwolscine from adrenergic alpha2C receptor | Bioorg Med Chem Lett 20: 3654-7 (2010) Article DOI: 10.1016/j.bmcl.2010.04.099 BindingDB Entry DOI: 10.7270/Q2474B1C | |||||||||||
More data for this Ligand-Target Pair |