Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Aurora kinase A (Homo sapiens (Human)) | BDBM50449313 (CHEMBL3125820) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.64E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Konkuk University Curated by ChEMBL | Assay Description Inhibition of human aurora A kinase using LRRASLG as substrate by scintillation counting in presence of [gamma-33P]ATP | Bioorg Med Chem 22: 1809-20 (2014) Article DOI: 10.1016/j.bmc.2014.01.058 BindingDB Entry DOI: 10.7270/Q21R6S1R | |||||||||||
More data for this Ligand-Target Pair |