Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bcl-2-like protein 1 (Homo sapiens (Human)) | BDBM50379281 (CHEMBL2011504) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 930 | n/a | n/a | n/a | n/a | n/a |
Broad Institute of Harvard and MIT Curated by ChEMBL | Assay Description Displacement of BakBH3 from Bcl-xL by DEL method | Bioorg Med Chem 20: 1979-89 (2012) Article DOI: 10.1016/j.bmc.2011.11.071 BindingDB Entry DOI: 10.7270/Q22J6CVS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-like protein 1 (Homo sapiens (Human)) | BDBM50379281 (CHEMBL2011504) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 930 | n/a | n/a | n/a | n/a | n/a |
University of Utah Curated by ChEMBL | Assay Description Binding affinity to human Bcl-xL after 1 hr by fluorescence polarization assay | J Med Chem 59: 6629-44 (2016) Article DOI: 10.1021/acs.jmedchem.5b01874 BindingDB Entry DOI: 10.7270/Q2N58QV5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-like protein 1 (Homo sapiens (Human)) | BDBM50379281 (CHEMBL2011504) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 930 | n/a | n/a | n/a | n/a | n/a |
University of Utah Curated by ChEMBL | Assay Description Binding affinity to human Bcl-xL after 1 hr by fluorescence polarization assay | J Med Chem 59: 6629-44 (2016) Article DOI: 10.1021/acs.jmedchem.5b01874 BindingDB Entry DOI: 10.7270/Q2N58QV5 | |||||||||||
More data for this Ligand-Target Pair |