Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM84342 (4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase KEGG PC cid PC sid PDB UniChem Similars | PubMed | n/a | n/a | n/a | 610 | n/a | n/a | n/a | n/a | n/a |
Merck, Sharp, and Dohme Research Laboratories | Assay Description The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP. | J Biol Chem 264: 13572-8 (1989) BindingDB Entry DOI: 10.7270/Q29G5KDJ | |||||||||||
More data for this Ligand-Target Pair |