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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50272103'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Cannabinoid receptor 2


(Homo sapiens (Human))
BDBM50272103
PNG
(CHEMBL499877 | N-(9-Ethyl-9H-carbazol-3-yl)-3-(3-p...)
Show SMILES CCn1c2ccccc2c2cc(NC(=O)CCc3nc(no3)-c3ccccc3)ccc12
Show InChI InChI=1S/C25H22N4O2/c1-2-29-21-11-7-6-10-19(21)20-16-18(12-13-22(20)29)26-23(30)14-15-24-27-25(28-31-24)17-8-4-3-5-9-17/h3-13,16H,2,14-15H2,1H3,(H,26,30)
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PC cid
PC sid
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Article
PubMed
n/an/an/an/a 150n/an/an/an/a



Amgen Inc.

Curated by ChEMBL


Assay Description
Agonist activity at human recombinant CB2 receptor expressed in Sf9 cells by GTP-europium binding assay


J Med Chem 51: 5019-34 (2008)


Article DOI: 10.1021/jm800463f
BindingDB Entry DOI: 10.7270/Q2W096VS
More data for this
Ligand-Target Pair