Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50330768 ((6aR,10aR)-1-bromo-6,6,9-trimethyl-3-(2-methylhept...) | PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 28 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Clemson University Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cells after 1 hr by liquid scintillation spectrophotometry | Bioorg Med Chem 18: 7809-15 (2010) Article DOI: 10.1016/j.bmc.2010.09.061 BindingDB Entry DOI: 10.7270/Q2ZK5HP7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50330768 ((6aR,10aR)-1-bromo-6,6,9-trimethyl-3-(2-methylhept...) | PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 28.6 | n/a | n/a | n/a | n/a |
Clemson University Curated by ChEMBL | Assay Description Agonist activity at human CB2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding after 1.5 hrs by liquid scintillation... | Bioorg Med Chem 18: 7809-15 (2010) Article DOI: 10.1016/j.bmc.2010.09.061 BindingDB Entry DOI: 10.7270/Q2ZK5HP7 | |||||||||||
More data for this Ligand-Target Pair |