Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50392710 (CHEMBL2151379) | PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 385 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Avenue de l'Universit£ Curated by ChEMBL | Assay Description Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting | Eur J Med Chem 58: 396-404 (2012) Article DOI: 10.1016/j.ejmech.2012.10.031 BindingDB Entry DOI: 10.7270/Q2474BZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50392710 (CHEMBL2151379) | PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 371 | n/a | n/a | n/a | n/a |
Avenue de l'Universit£ Curated by ChEMBL | Assay Description Agonist activity at human CB2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assay | Eur J Med Chem 58: 396-404 (2012) Article DOI: 10.1016/j.ejmech.2012.10.031 BindingDB Entry DOI: 10.7270/Q2474BZG | |||||||||||
More data for this Ligand-Target Pair |