Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Carboxypeptidase A1 (Bos taurus (bovine)) | BDBM50100009 (2-(1H-Imidazol-4-yl)-3-phenyl-propionic acid | 2-(...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 260 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pohang University of Science and Technology Curated by ChEMBL | Assay Description Inhibitory constant of carboxypeptidase A (CPA) in absence of Zinc ion. | Bioorg Med Chem Lett 11: 1425-7 (2001) BindingDB Entry DOI: 10.7270/Q2GX49VQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Carboxypeptidase A1 (Homo sapiens (Human)) | BDBM50100009 (2-(1H-Imidazol-4-yl)-3-phenyl-propionic acid | 2-(...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasma | J Med Chem 46: 5294-7 (2003) Article DOI: 10.1021/jm034141y BindingDB Entry DOI: 10.7270/Q27H1J0Z | |||||||||||
More data for this Ligand-Target Pair |